Exemestane is a new generation of drug that blocks enzymesresponsible for aromatisation. Exemestane is significantly differentfrom drugs belonging to the class of aromatase inhibitors.Exemestane is a better drug, Familiar aromatase inhibitors have onlya temporary efficiengy, but Exemestane has an irreversible andpermanent effect As a result of the drug are suppressed 85.9% ormore estrogens in the body of the athlete.
Exemestane during steroid cycle prevents the side effects thatsteroids can cause - flavoring. It should be noted that the effect of Exemestane is fundamentally different from the usual action of Nolvadex for many athletes. it is known that Tamoxifen has no effecton the aromatization process. It just begins to interact with thecellular estrogen receptors, preventing estrogen to join them andform a bond.
Exemestane also acts on the process of flavoring and suppressesit Exemestane structure is wery similar to a naturally occurringsteroid - androstenedione. Exemestane principle of operation is thatit irreversibly binds to active enzymes hormones. As a result.hormones lose their activity, Exemestane has no estrogenic orprogestogenic activity. But it is characterized by mild androgenicactivity.
Breast cancer in postmenopausal women (natural or induced).progressing against the background of antiestrogen therapy, non-steroidal aromatase inhibitors or progestins.
Dosage for men - 12.5-25 mg/day, dosage for Women - 12.5 mg/day
Exemestane side effects may occur frequently and in varyingdegrees. For example an athlete may face unpleasant consequencessuch as: nausea, fatique. sweating, dizziness, headache, skin rash.insomnia. etc.